Jadegoud Yaligar1, Rengaraj Anantharaj1, Giang Le Thi Thu 1, Ritu Chawla2, Sanjay Kumar Verma1, Venkatesh Gopalan1, Houchun H Hu3, Karthik Mallilankaraman2, and S. Sendhil Velan1
1Laboratory of Molecular Imaging, Singapore Bioimaging Consortium, Singapore, Singapore, 2Department of Physiology, National University of Singapore, Singapore, Singapore, 3Department of Radiology, Nationwide Children’s Hospital, Columbus, OH, United States
Synopsis
Understanding the functional aspects of BAT
under obese and overweight conditions is important to improve metabolic
dysfunction. Mechanisms that regulate the quality of BAT are influenced by
dietary lipids and plays a vital role in fat oxidation. Our imaging and
molecular biology data suggests that lipid oxidative capacity of the
mitochondria in iBAT is compromised with increased accumulation of lipids. High
fat dietary feeding did not affect the mitochondrial content. However, the mitochondrial
function was profoundly impaired. The novel finding in this study is the
reduction in the activity of complex II in HFD fed rats leading to
mitochondrial dysfunction.
Purpose
Investigation of mechanistic interlink between high fat diet induced
mitochondrial dysfunction and impaired lipid oxidation in brown adipose tissue.Introduction
Brown adipose
tissue (BAT) is involved in energy dissipation by thermogenic process that can
modulate fat oxidation under stimulated conditions1-3. Understanding
the functional aspects of BAT in response to HFD in obese and overweight
conditions is important. Mechanisms that regulate the quality of BAT were influenced
by dietary lipids and plays vital role in fat oxidation4. In this
study we investigated the mechanistic link between BAT mitochondrial
dysfunction and impaired lipid oxidation in response to high fat dietary
intervention.Methods
Animal studies were conducted as per the protocols approved by the
institutional animal care and use committee (A-star). Male Wistar rats at 7 weeks
of age were randomized into two groups and were fed with CD (n=6) and HFD (n=6)
diet until 15 weeks of age. Longitudinal MR data was acquired at 7, 11 and 15
weeks of age. Animals were imaged at thermoneutral temperature of
36±0.5 °C and later exposed to acute cold temperature of 18±0.5°C for 1hr. Experiments
were
performed using a 7T MRI scanner. Spectroscopy experiments were performed in iBAT
region TR;4s, TE;13ms, voxel;21mm3, Av;64. After terminal invivo experiments, BAT
samples were collected and tissue sections were stained for hematoxylin and
eosin staining. Western blot analysis was carried out on lysates from BAT
tissues collected. Complex activities were measured from mitochondria isolated
from BAT tissues. The mRNA analysis of UCP1 gene was performed on BAT and were
normalized to beta actin.Results and Discussion
HFD group rats were insulin resistant by 11 weeks. Figure 1A shows the fat
fraction image with a voxel placed in iBAT region. Figures
1B,C,D, E and F show the invivo
spectra from iBAT and Figure-1G shows the fat content at thermoneutral and cold exposed condition.
At thermoneutral condition the lipid content in iBAT significantly increased
for HFD groups. Under cold exposed condition, reduction of fat content for
CD fed rats at 7, 11 and 15 weeks was 28.72±1.02%, 16.46%±0.98% and 13.95± 1.13% respectively. For HFD group the
reduction of fat at 11w was 12.35±1.08% (P<0.05)
and at 15 weeks the fat content did not change significantly in response to acute cold induced BAT
activation. Thermogenic function of activated BAT requires the utilization of
fatty acids as substrates, leading to uncoupling of protein 1 (UCP1) in
mitochondrial membrane. UCP1 (Figure 2A) expression at 11 weeks was increased
significantly for HFD group compared to CD group, indicating the metabolic
adaptation associated with the compensatory response of mitochondria in
response to HFD overload. At
15 weeks, the UCP1 in iBAT of HFD group failed to show this adaptive increase
in expression. To further evaluate the oxidizing capacity of iBAT in HFD rats, we studied the expression of CPT1 (Figure 2B,C). In HFD group the CPT1
expression reduced at 15 weeks compared to 11 weeks, indicating the compromised
mitochondrial efficiency to oxidize the lipids and is consensus with UCP1
results. We identified the compromised enzyme activity of complex II in iBAT
tissues of HFD group. Figures 3A,B,C show Immunoblot analysis and
quantification of complex II subunits (SDHA and SDHB) in CD and HFD groups. Complex
II enzyme activity (Figure 4A, B) was significantly lower in 11 and 15 weeks
old HFD group compared to CD group. Our data suggests that with HFD feeding the
mitochondrial content was not affected (Figure 3B,C), however the mitochondrial
functionality (Figure 4A,B) was profoundly compromised by HFD feeding. The ROS is essential for iBAT mitochondria and it was significantly decreased in
HFD group (Figure-4C). Defective complex II activity reduces the
reverse electron transport mediated mitochondrial ROS production which is
crucial for BAT mitochondria to activate UCP1. The net effect is down
regulation of UCP1 and impaired thermogenesis is mechanistically showed in Figure 5A, B.
Conclusions
Our data suggests that lipid oxidative capacity of the mitochondria in
iBAT was compromised with increased accumulation of lipids. HFD feeding did not
affect the mitochondrial content. However, the mitochondrial functionality was profoundly
impaired. Novel finding in our study is reduction in the activity of
complex II in HFD group leading to mitochondrial dysfunction. Defective
complex II activity reduces the reverse electron transport mediated mitochondrial
ROS production at Complex I and Complex III sites which is crucial for BAT
mitochondria to activate UCP1 by sulfenylation of UCP1 Cys253 site. Although the UCP1 expression in HFD rats at 15
weeks did not get altered, the activity of UCP1 was down regulated by defective
Complex II activity that deprived iBAT from the essential mitochondrial ROS.
Our results on defective Complex II mediated decreased UCP1 activity correlates
with decreased lipid oxidation observed by MRS.Acknowledgements
No acknowledgement found.References
- Pradhan A, Obesity, metabolic syndrome,
and type 2 diabetes: inflammatory basis of glucose metabolic disorders, Nutr
Rev. 2007;65(12 Pt 2):S152-6.
- Kristy L, Townsend, et al, Brown Fat Fuel
Utilization and Thermogenesis, Trends Endocrinol Metab, 2014 ;25(4):168–177.
- Harms M, et al, Brown and beige
fat: development, function and therapeutic potential, Nat Med, 2013; 19(10):1252-63.
- Calderon-Dominguez, M., Fatty acid
metabolism and the basis of brown adipose tissue function, Adipocyte, 2016; 5: 98-118.