Akira Sumiyoshi1,2, Satoshi Ikemoto1, Elliot A. Stein1, Yihong Yang1, and Hanbing Lu1
1National Institute on Drug Abuse, National Institutes of Health, Baltimore, MD, United States, 2National Institutes for Quantum and Radiological Science and Technology, Chiba, Japan
Synopsis
Although resting-state functional MRI (rs-fMRI) is extensively used to
study brain circuitry, recent animal studies suggest a non-neuronal origin of
the rs-fMRI signal. We hypothesized that astrocytes may play an important role
in rs-fMRI signal. We used chemogenetic technology to selectively activate
astrocytes (increasing Ca2+ levels) and recorded rs-fMRI signals in lightly
anesthetized rats. Chemogenetic activation of astrocytes following 0.1 mg/kg of clozapine injection induced signal intensity changes and reduced functional
connectivity. These in vivo results are consistent with previous brain slice
studies, confirming a potentially important role of astrocytes in rs-fMRI
signals.
Introduction
Resting-state functional MRI (rs-fMRI) is a neuroimaging method that
assesses the strength of functional interactions between brain regions when a
subject is not engaged in an explicit task. We have previously identified a
robust rs-fMRI circuit between the left and right striatum in lightly anesthetized
rats.
1 However, simultaneously recorded local field potentials (LFPs)
and rs-fMRI signals were only weakly correlated (
r < 0.1). A recent optical imaging study in awake mice also reported
weak correlations between LFPs and hemodynamic signals during periods of “true”
rest in the absence of external stimuli and body movements.
2 These
results suggest a non-neuronal origin of the rs-fMRI signal. Astrocytes, a type
of glial cell, are essential for the supply of energy metabolites to neurons
and, by means of their endfoot processes, provide a physical link to the
vasculature. We thus hypothesized that astrocytes may directly regulate the vasculature
and may play an important role in mediating neurovascular coupling. The aim of
this study is to investigate the role of astrocytes in rs-fMRI signal using chemogenetic
technology (DREADD; designer receptors exclusively activated by designer drugs).
Specifically, we explored the effects of astrocyte-specific DREADD enhancement
of calcium activity in striatal astrocytes on the rs-fMRI signal.
Methods
In 12 male Sprague-Dawley rats (373–541 g), the active DREADD AAV5-GFAP-hM3D(Gq)-mCherry
was microinjected unilaterally into the striatum while AAV5-GFAP-eGFP was
microinjected as a control into the contralateral striatum (Fig. 1A). The virus
vectors were obtained from Duke Viral Vector Core.3 Left and right sides
were counter-balanced across subjects. After three weeks period for the expression
of DREADD receptors, multiple DREADD-fMRI recordings were conducted from the
same subjects with a one-week interval between data acquisitions (Fig. 1B). Clozapine
(0.1 or 0.5 mg/kg) or clozapine N-oxide (3.0 mg/kg) was used as DREADD agonists.4 Rs-fMRI signals (TR = 1.5 s and spatial resolution =
0.547 x 0.547 x 1 mm3) were acquired using a 9.4-T MRI system with a
20-mm diameter surface coil. Rats were lightly anesthetized with 0.02 mg/kg/hr of
Dexmedetomidine and 0.5% of Isoflurane. All procedures were approved by the
NIDA-IRP Animal Care and Use Committee.Results
The selective expression of DREADD receptors in striatal astrocytes were
confirmed using immunohistochemistry (Fig. 1C and D). Region-of-interest (ROI) analyses
of rs-fMRI signals, based on individual postmortem histological images (Fig.
2A), demonstrated that astrocyte DREADD activation using 0.1 mg/kg of clozapine
induced intensity changes in the rs-fMRI signal that started about 2 min after
drug administration and lasted for approximately 20 min (Fig. 2B). In contrast,
no changes in signal were seen following 0.5 mg/kg of clozapine or 3.0 mg/kg of clozapine N-oxide injection (Fig. 2C). At the group level there was a
significant difference in mean rs-fMRI signal (p < 0.001) between the DREADD and control side ROIs (Fig. 3A). The
rs-fMRI signals after DREADD activation showed a bi-phasic response without a
few exceptions that showed only an increase or decrease response (Fig. 3B). The
rs-fMRI connectivity strength between the DREADD and control side ROIs was significantly
reduced after unilateral DREADD activation (one-way ANOVA, p < 0.01) (Fig. 3C).Discussion
Previous brain slice experiments
demonstrated that astrocytes are capable of dilating and constricting adjacent
arterioles depending on the Ca2+ level of astrocytic endfoot processes
and activation of Ca2+ dependent BK channels.5 Brain
slice experiments also demonstrate that astrocytes produce a variety of vasodilators
and vasoconstrictors (e.g. prostaglandins, epoxyeicosatrienoic acids, and 20-hydroxyeicosatetraenoic
acids) via an increase of intracellular Ca2+ levels.6 The
rs-fMRI results demonstrated herein using cell-specific DREADD technology are consistent
with these previous slice studies, confirming a potentially bidirectional role
of astrocytes in generating the rs-fMRI signal.7 Several technical
issues need to be considered. First, the rs-fMRI results were not consistent
across subjects (Fig. 3B), suggesting differences in cells that were infected
and their local circuits, different number of cells, different state of
anesthesia, or ongoing brain processes as modulated from other brain regions
and circuits. Second, the direct in vivo relationships between astrocytic Ca2+
levels and rs-fMRI signals were not measured, making difficult to infer the
temporal dynamics of astrocytic Ca2+ levels compared with rs-fMRI signals.
Further technical refinements will be required in the future study.Conclusion
We demonstrated a causal relationship between astrocytic activation and
rs-fMRI signals using chemogenetic technology. Upon the selective activation of
astrocytes, rs-fMRI signals were fluctuated and the functional connectivity between
hemispheres was perturbed. However, several technical issues need to be
addressed in the future study to further investigate the role of astrocytes in rs-fMRI
signal.Acknowledgements
This work was supported by the Japan Society for the Promotion of
Science Overseas Research Fellowships (to AS) and the Intramural Research
Program of the National Institute on Drug Abuse, NIH.References
- Jaime S, Gu H, Sadacca BF,
et al. Delta rhythm orchestrates the neural activity underlying the resting state
BOLD signal via phase-amplitude coupling. Cereb. Cortex, in press.
- Winder AT, Echagarruga C,
Zhang Q, et al. Weak correlations between hemodynamic signals and ongoing
neural activity during the resting state. Nat. Neurosci. 2017; 20 (12):
1761–1769.
-
Bull C, Freitas KCC, Zou
S, et al. Rat nucleus accumbens core astrocytes modulate reward and the
motivation to self-administer ethanol after abstinence. Neuropsychopharmacology
2014; 39 (12), 2835–2845.
-
Gomez JL, Bonaventura J,
Lesniak W, et al. Chemogenetics revealed: DREADD occupancy and activation via
converted clozapine. Science 2017; 357 (6350), 503–507.
-
Girouard H, Bonev AD,
Hannah RM, et al. Astrocytic endfoot Ca2+ and BK channels determine
both arteriolar dilation and constriction. Proc. Natl. Acad. Sci. U.S.A. 2010; 107
(8), 3811–3816.
-
Attwell D, Buchan AM,
Charpak S, et al. Glial and neuronal control of brain blood flow. Nature 2010; 468
(7321): 232–243.
-
Gordon GRJ, Howarth C,
MacVicar BA. Bidirectional control of blood flow by astrocytes: A role for tissue
oxygen and other metabolic factors. Adv. Exp. Med. Biol. 2016; 903, 209–219.